Acetylene functionalized BODIPY dyes and their application in the synthesis of activity based proteasome probes.

نویسندگان

  • Martijn Verdoes
  • Ulrik Hillaert
  • Bogdan I Florea
  • Myra Sae-Heng
  • Martijn D P Risseeuw
  • Dmitri V Filippov
  • Gijsbert A van der Marel
  • Herman S Overkleeft
چکیده

The synthesis of three acetylene functionalized BODIPY dyes is described. These dyes are used to fluorescently modify an azido functionalized epoxomicin analogue employing the Huisgen 1,3-dipolar cycloaddition, resulting in a panel of fluorescent epoxomicin derived proteasome probes.

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عنوان ژورنال:
  • Bioorganic & medicinal chemistry letters

دوره 17 22  شماره 

صفحات  -

تاریخ انتشار 2007